Extending Pummerer reaction chemistry. Application to the oxidative cyclization of tryptophan derivatives.
Journal
  Organic letters.
Citation
  Org Lett. 6(17):2849-52
Publication date
  2004 Aug 19
Authors
  Feldman KS
Karatjas AG
Grant agencies
  National Institute of General Medical Sciences
Grants
  NIGMS GM35727
Abstract
  The diastereoselective oxidative cyclization of a beta-oxygenated tryptophan derivative is reported. This process, which utilizes a new variant of the Pummerer reaction, may have application in TMC-95A synthesis.